Cart
sales@molnova.com
Calcium channel-modulator-1
CAS No. 136941-70-3
Calcium channel-modulator-1( —— )
Catalog No. M32746 CAS No. 136941-70-3
Calcium channel-modulator-1, a calcium channel-modulator (IC50: 0.8 μM), specializes in blocking aortic constriction.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 211 | Get Quote |
|
| 5MG | 258 | Get Quote |
|
| 10MG | 416 | Get Quote |
|
| 25MG | 685 | Get Quote |
|
| 50MG | 908 | Get Quote |
|
| 100MG | 1251 | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
-
Product NameCalcium channel-modulator-1
-
NoteResearch use only, not for human use.
-
Brief DescriptionCalcium channel-modulator-1, a calcium channel-modulator (IC50: 0.8 μM), specializes in blocking aortic constriction.
-
DescriptionCalcium channel-modulator-1 is a calcium channel modulator; blocks aortic contraction with an IC50 of 0.8 μM.
-
In Vitro——
-
In VivoOral administration of Calcium channel-modulator-1 (20 mg/kg) causes a 35-37% decrease in systolic blood pressure in spontaneously hypertensive rats. However, iv administration of Calcium channel-modulator-1 to anesthetized spontaneously hypertensive rats causes a decrease in blood pressure which was more pronounced and long-lasting than that of nifedipine.
-
Synonyms——
-
PathwayGPCR/G Protein
-
TargetCalcium Channel
-
RecptorCalcium Channel
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number136941-70-3
-
Formula Weight579.45
-
Molecular FormulaC26H24Cl2N2O7S
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESC(OCCCN1S(=O)(=O)C=2C(C1=O)=CC=CC2)(=O)C=3C(C(C(OC)=O)=C(C)NC3C)C4=C(Cl)C(Cl)=CC=C4
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Sunkel CE, et al. Synthesis of 3-[(2,3-dihydro-1,1,3-trioxo-1,2-benzisothiazol-2-yl)alkyl] 1,4-dihydropyridine-3,5-dicarboxylate derivatives as calcium channel modulators. J Med Chem. 1992 Jun 26;35(13):2407-14.?
molnova catalog
related products
-
Pranidipine
Pranidipine is a novel, long-acting 1,4-dihydropyridine calcium channel blocker.
-
Lanthanum(III) chlor...
Lanthanum(III) chloride is an inorganic compound which used in biochemical research to block the activity of divalent cation channels, especially calcium channels.
-
1-(aminomethyl)cyclo...
1-(aminomethyl)cyclopropanecarboxylic acid hydrochloride inhibits L amino acid transporter proteins and the α2δ subunit of voltage-gated calcium channels.
